SCHEMBL19954966

SCHEMBL19954966

COC(=O)[C@]1(C)CCCN1C(=O)I

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.35
MEN1 O00255 1/20 0.33
CYP3A4 P08684 1/20 0.33
KMT2A Q03164 1/20 0.33
USP2 O75604 1/20 0.32
PIK3CA P42336 2/20 0.31
CYP4F2 P78329 1/20 0.30
CYP4A11 Q02928 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2044620 0.84 NPSR1 (0.36) NPSR1MEN1CYP3A4KMT2AUSP2
SCHEMBL18352400 0.84 MEN1 (0.41) NPSR1MEN1CYP3A4KMT2A
SCHEMBL15214890 0.79 NPSR1 (0.37) NPSR1MEN1CYP3A4KMT2AUSP2
SCHEMBL12385681 0.79 DPP4 (0.34) NPSR1MEN1CYP3A4KMT2AUSP2
SCHEMBL15214887 0.78 CYP3A4 (0.37) NPSR1MEN1CYP3A4KMT2ACYP4F2
SCHEMBL3000664 0.77 GRIN2B (0.40) USP2
SCHEMBL3000663 0.77 GRIN2B (0.40) USP2
SCHEMBL10039817 0.77 GRIN2B (0.40) USP2
SCHEMBL12934881 0.76 GAA (0.40)
SCHEMBL23643970 0.76 NPSR1 (0.38) NPSR1MEN1CYP3A4KMT2AUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9914721-B2 Use of benzimidazole-proline derivatives IDORSIA PHARMACEUTICALS LTD (CH) 2018-03-13 US disclosed