SCHEMBL19957396

SCHEMBL19957396

C[C@H]1CCCN(c2ccc(C#N)c3ncccc23)C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 6/20 0.53
TLR9 Q9NR96 6/20 0.51
TLR7 Q9NYK1 6/20 0.51
AR P10275 6/20 0.45
LRRK2 Q5S007 1/20 0.43
KDM4E B2RXH2 2/20 0.42
NPC1 O15118 1/20 0.42
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
CASP1 P29466 1/20 0.42
RAB9A P51151 1/20 0.42
CASP7 P55210 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
KCNMA1 Q12791 1/20 0.40
CTSB P07858 1/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21795290 0.93 TLR8 (0.54) TLR8TLR9TLR7ARKDM4E
SCHEMBL17840412 0.87 TLR8 (0.65) TLR8TLR9TLR7AR
SCHEMBL17840411 0.87 TLR8 (0.65) TLR8TLR9TLR7AR
SCHEMBL21661053 0.85 TLR9 (0.53) TLR8TLR9TLR7ARLRRK2
SCHEMBL4876295 0.84 AR (0.63) TLR8TLR9TLR7ARKDM4E
SCHEMBL30317631 0.82 MAPT (0.44) TLR7KDM4ENPC1ALDH1A1GAA
SCHEMBL26351021 0.82 TLR8 (0.62) TLR8TLR9TLR7ARKCNMA1
SCHEMBL23415867 0.81 TLR9 (0.63) TLR8TLR9TLR7AR
SCHEMBL21795382 0.81 TLR8 (0.54) TLR8TLR9TLR7ARKDM4E
SCHEMBL21795300 0.81 TLR8 (0.52) TLR8TLR9TLR7ARKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057948-B1 SELECTIVELY SUBSTITUTED QUINOLINE DERIVATIVES EISAI R&D MAN CO LTD (JP) 2018-03-14 EP disclosed