SCHEMBL19959568

SCHEMBL19959568

CCOC(=O)C(OC[C@H]1O[C@@H](n2cnc3c(NC(=O)OC(C)(C)C)nc(Cl)nc32)C(N=[N+]=[N-])[C@@H]1O)C(=O)OCC

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NT5E P21589 15/20 0.68
CD99 P14209 1/20 0.44
ADORA3 P0DMS8 2/20 0.43
ADORA1 P30542 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19949327 0.86 NT5E (0.51) NT5ECD99ADORA3
SCHEMBL20333709 0.85 NT5E (0.56) NT5E
SCHEMBL30262574 0.85 NT5E (0.56) NT5E
SCHEMBL19961924 0.84 NT5E (0.48) NT5ECD99ADORA3
SCHEMBL30262553 0.81 NT5E (0.71) NT5ECD99ADORA1
SCHEMBL19948958 0.81 NT5E (1.00) NT5ECD99
SCHEMBL19949062 0.81 NT5E (1.00) NT5ECD99
SCHEMBL30262580 0.81 NT5E (1.00) NT5ECD99
SCHEMBL19948652 0.81 NT5E (1.00) NT5ECD99
SCHEMBL30262592 0.81 NT5E (1.00) NT5ECD99

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018049145-A1 ECTONUCLEOTIDASE INHIBITORS AND METHODS OF USE THEREOF CALITHERA BIOSCIENCES, INC. (US) 2018-03-15 WO disclosed