SCHEMBL19966583

SCHEMBL19966583

Cc1nc2c(F)cc(-c3nc(Nc4cccc(C(=O)N5CCC(N(C)C)C5)n4)ncc3F)cc2n1C(C)C

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.63
CDK6 Q00534 18/20 0.63
CDK2 P24941 15/20 0.63
CDK1 P06493 7/20 0.59
CDK9 P50750 5/20 0.59
CDK7 P50613 4/20 0.59
CCNB1 P14635 4/20 0.59
CCNE1 P24864 4/20 0.59
CCND1 P24385 3/20 0.57
CCND3 P30281 3/20 0.57
CDK5 Q00535 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17488764 0.88 CDK4 (0.71) CDK4CDK6CDK2CDK1CDK9
SCHEMBL17488816 0.88 CDK4 (0.71) CDK4CDK6CDK2CDK1CDK9
SCHEMBL17477127 0.88 CDK4 (0.71) CDK4CDK6CDK2CDK1CDK9
SCHEMBL19966468 0.86 CDK4 (0.61) CDK4CDK6CDK2CDK1CDK9
SCHEMBL28560439 0.86 CDK4 (0.60) CDK4CDK6CDK2CDK1CDK9
SCHEMBL19966526 0.85 CDK4 (0.67) CDK4CDK6CDK2CDK1CDK9
SCHEMBL17488869 0.84 CDK4 (0.66) CDK4CDK6CDK2CDK1CDK9
SCHEMBL19966465 0.83 CDK4 (0.64) CDK4CDK6CDK2CDK1CDK9
SCHEMBL17489102 0.83 CDK4 (0.64) CDK4CDK6CDK2CDK1CDK9
SCHEMBL19968123 0.82 CDK4 (0.61) CDK4CDK6CDK2CDK1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018045957-A1 CDK4/6 INHIBITOR AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 江苏豪森药业集团有限公司 2018-03-15 WO disclosed