SCHEMBL19968024

SCHEMBL19968024

Cc1nc(Nc2ncc(F)c(-c3ccc4nc(C)n(C(C)C)c4c3)n2)ccc1C(=O)N1CCCN(C)CC1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 12/20 0.58
CDK2 P24941 9/20 0.55
CDK1 P06493 9/20 0.55
PIM1 P11309 1/20 0.51
CDK4 P11802 12/20 0.51
CCNB1 P14635 5/20 0.51
CCNE1 P24864 5/20 0.51
CDK9 P50750 4/20 0.51
CDK7 P50613 3/20 0.51
HDAC1 Q13547 1/20 0.51
DYRK2 Q92630 2/20 0.50
CCND1 P24385 1/20 0.50
CCND3 P30281 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19968032 0.90 CDK4 (0.63) CDK6CDK2CDK1CDK4CCNB1
SCHEMBL19968106 0.87 CDK6 (0.51) CDK6CDK2CDK1PIM1CDK4
SCHEMBL19968053 0.87 CDK6 (0.52) CDK6CDK2CDK1PIM1CDK4
SCHEMBL30789752 0.87 CDK6 (0.52) CDK6CDK2CDK1PIM1CDK4
SCHEMBL19968038 0.84 CDK4 (0.64) CDK6CDK2CDK1CDK4CCNB1
SCHEMBL19968108 0.84 CDK6 (0.51) CDK6CDK2CDK1PIM1CDK4
SCHEMBL17488982 0.83 CDK6 (0.69) CDK6PIM1DYRK2CCND1
SCHEMBL19968040 0.81 CDK4 (0.66) CDK6CDK2CDK1PIM1CDK4
SCHEMBL17489295 0.81 CDK6 (0.79) CDK6PIM1DYRK2CCND1
SCHEMBL19968116 0.80 CDK4 (0.64) CDK6CDK2CDK1PIM1CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018045956-A1 BENZIMIDAZOLE COMPOUND KINASE INHIBITOR, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 江苏豪森药业集团有限公司 2018-03-15 WO disclosed