SCHEMBL19968054

SCHEMBL19968054

Cc1nc(Nc2ncc(F)c(-c3cc(F)c4nc(C)n(C(C)C)c4c3)n2)ccc1C(=O)N1CCC(N2CCC2)CC1

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.62
CDK1 P06493 12/20 0.62
CCNB1 P14635 10/20 0.62
CCNE1 P24864 10/20 0.62
CDK6 Q00534 13/20 0.60
CDK2 P24941 12/20 0.60
CDK9 P50750 5/20 0.59
CCNT1 O60563 1/20 0.59
CCND3 P30281 1/20 0.59
CDK7 P50613 3/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19968086 0.98 CDK4 (0.61) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL29406457 0.98 CDK4 (0.61) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL19968063 0.94 CDK4 (0.60) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL19968045 0.92 CDK4 (0.61) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL19967978 0.90 CDK4 (0.60) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL19968061 0.90 CDK4 (0.60) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL30926189 0.90 CDK4 (0.61) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL19968031 0.90 CDK4 (0.61) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL19968047 0.90 CDK4 (0.59) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL19967982 0.90 CDK4 (0.60) CDK4CDK1CCNB1CCNE1CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018045956-A1 BENZIMIDAZOLE COMPOUND KINASE INHIBITOR, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 江苏豪森药业集团有限公司 2018-03-15 WO disclosed