SCHEMBL19973036

SCHEMBL19973036

COc1cccc(COC(N)=O)c1OC

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.48
ABCB1 P08183 2/20 0.48
ABCG2 Q9UNQ0 1/20 0.48
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA14 Q9ULX7 1/20 0.48
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
LMNA P02545 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
KDM4E B2RXH2 1/20 0.47
CYP1A2 P05177 1/20 0.47
MAPT P10636 2/20 0.46
ALDH1A1 P00352 1/20 0.46
HIF1A Q16665 1/20 0.46
ATM Q13315 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2341243 0.87 ABCB1 (0.50) RXFP1ABCB1ABCG2CA12CA1
SCHEMBL13034146 0.85 RXFP1 (0.49) RXFP1ABCB1ABCG2CA12CA1
SCHEMBL113807 0.85 IDO1 (0.59) KMT2AMEN1LMNASMN1; SMN2KDM4E
SCHEMBL28769967 0.84 KMT2A (0.50) RXFP1ABCB1ABCG2CA12CA1
SCHEMBL29272775 0.83 KMT2A (0.43) KMT2AMEN1LMNASMN1; SMN2KDM4E
SCHEMBL4684928 0.81 CA12 (0.55) ABCB1ABCG2CA12CA1CA2
SCHEMBL490497 0.80 KMT2A (0.47) RXFP1ABCB1ABCG2CA12CA1
SCHEMBL7596038 0.80 ABCB1 (0.46) RXFP1ABCB1ABCG2KMT2AMEN1
SCHEMBL1032325 0.80 CA12 (0.50) ABCB1ABCG2CA12CA1CA2
SCHEMBL4369269 0.77 ABCB1 (0.57) ABCB1ABCG2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4323377-A1 VACCINES Adjuvance Technologies, Inc. (US) 2024-02-21 EP disclosed
WO-2023146892-A1 BIPHENYL-SUBSTITUTED EPITHELIAL SODIUM CHANNEL BLOCKING COMPOUNDS PARION SCIENCES, INC. (US) 2023-08-03 WO disclosed
WO-2023146896-A1 BICYCLIC-SUBSTITUTED EPITHELIAL SODIUM CHANNEL BLOCKING COMPOUNDS PARION SCIENCES, INC. (US) 2023-08-03 WO disclosed
WO-2023049218-A1 DOUBLE STRANDED OLIGONUCLEOTIDE COMPOSITIONS AND METHODS RELATING THERETO WAVE LIFE SCIENCES LTD. (SG) 2023-03-30 WO disclosed
WO-2022256480-A1 ARYLCOUMARIN SYNTHESIS WITH AZEOTROPIC REMOVAL OF WATER CONAGEN INC. (US) 2022-12-08 WO disclosed
EP-4061425-A1 DIRECTED CONJUGATION TECHNOLOGIES Kleo Pharmaceuticals, Inc. (US) 2022-09-28 EP disclosed
EP-3993818-A2 CD38-BINDING AGENTS AND USES THEREOF Kleo Pharmaceuticals, Inc. (US) 2022-05-11 EP disclosed
WO-2021234459-A9 DOUBLE STRANDED OLIGONUCLEOTIDE COMPOSITIONS AND METHODS RELATING THERETO WAVE LIFE SCIENCES LTD. (SG) 2022-02-03 WO disclosed
CN-107148453-B Photocurable composition 思美定株式会社 2021-08-17 CN disclosed
WO-2021102052-A1 DIRECTED CONJUGATION TECHNOLOGIES KLEO PHARMACEUTICALS, INC. (US) 2021-05-27 WO disclosed
CN-112805311-A Curable composition, cured product, and method for producing cured product 学校法人东京理科大学 2021-05-14 CN disclosed
CN-108431157-B Bonding method using photocurable adhesive 思美定株式会社 2021-02-05 CN disclosed
WO-2021003050-A2 CD38-BINDING AGENTS AND USES THEREOF KLEO PHARMACEUTICALS, INC. (US) 2021-01-07 WO disclosed
CN-105392845-B Photocurable composition 思美定株式会社 2020-10-20 CN disclosed
CN-111201295-A Photocurable adhesive composition and bonding method 思美定株式会社 2020-05-26 CN disclosed
EP-3630199-A1 OLIGONUCLEOTIDE COMPOSITIONS AND METHODS OF USE THEREOF Wave Life Sciences Ltd. (SG) 2020-04-08 EP disclosed
CN-107532061-B Pressure-sensitive adhesive 思美定株式会社 2020-03-03 CN disclosed
WO-2018223056-A1 OLIGONUCLEOTIDE COMPOSITIONS AND METHODS OF USE THEREOF WAVE LIFE SCIENCES LTD. (SG) 2018-12-06 WO disclosed
WO-2018053373-A1 USES OF SATL-INDUCIBLE KINASE (SIK) INHIBITORS FOR TREATING OSTEOPOROSIS THE GENERAL HOSPITAL CORPORATION (US) 2018-03-22 WO disclosed