SCHEMBL19976813

SCHEMBL19976813

O=C(/N=C(\Nc1n[nH]c2cc(C(F)(F)F)ccc12)NC1CCOCC1)c1ccc(Cl)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 4/20 0.47
GSK3B P49841 3/20 0.42
CRHR1 P34998 8/20 0.42
TRPA1 O75762 2/20 0.38
MAPK1 P28482 1/20 0.38
MAP2K4 P45985 1/20 0.38
MAPK6 Q16659 1/20 0.38
MAPKAPK5 Q8IW41 1/20 0.38
KIT P10721 1/20 0.38
FLT3 P36888 1/20 0.38
TRPV1 Q8NER1 1/20 0.38
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19976752 0.93 HDAC6 (0.49) HDAC6GSK3BCRHR1TRPA1MAPK1
SCHEMBL19976754 0.83 HDAC6 (0.52) HDAC6GSK3BTRPA1MAPK1MAP2K4
SCHEMBL19976829 0.82 HDAC6 (0.51) HDAC6GSK3BTRPA1MAPK1MAP2K4
SCHEMBL9921025 0.81 HDAC6 (0.39) HDAC6GSK3BMAPK1TRPV1KCNH2
SCHEMBL19976729 0.80 HDAC6 (0.49) HDAC6GSK3BCRHR1TRPA1MAPK1
SCHEMBL19976816 0.78 MAPT (0.46) HDAC6GSK3BMAPK1KITFLT3
SCHEMBL19976907 0.78 GSK3B (0.49) HDAC6GSK3BCRHR1TRPA1MAPK1
SCHEMBL19976733 0.78 HDAC6 (0.47) HDAC6GSK3BCRHR1TRPA1MAPK1
SCHEMBL19976753 0.78 GSK3B (0.47) HDAC6GSK3BCRHR1TRPA1MAPK1
SCHEMBL18558398 0.76 DYRK1A (0.37) HDAC6GSK3BMAPK1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9920012-B2 Indazole guanidine F1F0-ATPase inhibitors and therapeutic uses thereof LYCERA CORPORATION (US) 2018-03-20 US disclosed