SCHEMBL19979811

SCHEMBL19979811

C=CCOC(=O)N1CCC[C@@H]1c1nc(CNC(=O)CCCCCCCCNC(=O)COc2ccccc2C(=O)OC)no1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 18/20 0.38
HCRTR2 O43614 18/20 0.38
PRCP P42785 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19979812 1.00 HCRTR1 (0.38) HCRTR1HCRTR2PRCPALDH1A1TSHR
SCHEMBL19979730 0.83 HCRTR1 (0.36) HCRTR1HCRTR2ALDH1A1TSHR
SCHEMBL19975452 0.82 HCRTR1 (0.42) HCRTR1HCRTR2ALDH1A1TSHR
SCHEMBL19975485 0.82 HDAC8 (0.38) HCRTR1HCRTR2ALDH1A1TSHR
SCHEMBL19975484 0.82 HDAC8 (0.38) HCRTR1HCRTR2ALDH1A1TSHR
SCHEMBL19979742 0.81 CYP3A4 (0.39) PRCPALDH1A1TSHR
SCHEMBL19979749 0.81 CYP3A4 (0.39) PRCPALDH1A1TSHR
SCHEMBL19979810 0.80 DPP4 (0.35) ALDH1A1
SCHEMBL19979731 0.80 HCRTR1 (0.39) HCRTR1HCRTR2
Hydrochloric Acid SCHEMBL19975451 0.79 HCRTR1 (0.39) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053302-A1 MACROCYCLIC COMPOUNDS FOR THE INHIBITION OF INDOLEAMINE-2,3-DIOXYGENASE ACTIVITY AND USE THEREOF ENSEMBLE THERAPEUTICS CORPORATION (US) 2018-03-22 WO disclosed