SCHEMBL19981831

SCHEMBL19981831

CCC[C@H](N)C(=O)N1CCCCC1C

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 13/20 0.61
DPP7 Q9UHL4 13/20 0.55
DPP8 Q6V1X1 8/20 0.51
DPP9 Q86TI2 7/20 0.51
FAP Q12884 5/20 0.51
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12709891 0.87 DPP7 (0.59) DPP4DPP7DPP8DPP9FAP
SCHEMBL18774976 0.81 DPP4 (0.61) DPP4DPP7DPP8DPP9FAP
SCHEMBL18774982 0.81 DPP4 (0.61) DPP4DPP7DPP8DPP9FAP
Hydrochloric Acid SCHEMBL11171586 0.81 DPP4 (0.57) DPP4DPP7DPP8DPP9FAP
SCHEMBL7939898 0.80 DPP4 (0.66) DPP4DPP7DPP8DPP9FAP
SCHEMBL12938959 0.79 DPP7 (0.49) DPP4DPP7DPP8DPP9FAP
SCHEMBL24323544 0.78 DPP4 (0.63) DPP4DPP7DPP8DPP9FAP
SCHEMBL17814291 0.78 DPP4 (0.65) DPP4DPP7DPP8DPP9FAP
SCHEMBL12709872 0.77 DPP7 (0.46) DPP4DPP7DPP8DPP9FAP
SCHEMBL30314724 0.77 DPP4 (0.63) DPP4DPP7DPP8DPP9FAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512832-B1 TETRAHYDROISOQUINOLINE KAPPA OPIOID ANTAGONISTS RES TRIANGLE INST (US) 2021-05-19 EP disclosed
WO-2018053222-A1 TETRAHYDROISOQUINOLINE KAPPA OPIOID ANTAGONISTS RESEARCH TRAINGLE INSTITUTE (US) 2018-03-22 WO disclosed