SCHEMBL19986934

SCHEMBL19986934

FC(F)(F)Oc1cccc(-c2cnn3ccc(N4CCCCC4)nc23)c1

nearest known ligand 0.76

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 16/20 0.76
PIM2 Q9P1W9 12/20 0.76
FLT3 P36888 1/20 0.57
KCNH2 Q12809 1/20 0.56
SMPD3 Q9NY59 3/20 0.48
TGFBR2 P37173 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16210798 0.87 PIM1 (1.00) PIM1PIM2FLT3KCNH2
SCHEMBL102618 0.87 PIM1 (1.00) PIM1PIM2FLT3KCNH2
SCHEMBL14653595 0.80 PIM1 (0.63) PIM1PIM2FLT3KCNH2TGFBR2
SCHEMBL102845 0.80 PIM1 (0.60) PIM1PIM2FLT3KCNH2TGFBR2
SCHEMBL18362768 0.80 PIM1 (0.78) PIM1PIM2SMPD3
SCHEMBL1443512 0.79 SMPD3 (0.62) PIM1PIM2SMPD3
SCHEMBL19986964 0.78 PIM1 (0.83) PIM1PIM2FLT3KCNH2
SCHEMBL22421461 0.75 PIM1 (0.54) PIM1PIM2FLT3KCNH2TGFBR2
SCHEMBL4330227 0.75 PIM1 (0.65) PIM1PIM2FLT3KCNH2TGFBR2
SCHEMBL19494008 0.74 SMPD3 (0.56) PIM1PIM2SMPD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3812387-A1 HETEROCYCLIC PROTEIN KINASE INHIBITORS Sumitomo Dainippon Pharma Oncology, Inc. (US) 2021-04-28 EP disclosed
EP-3409278-B1 HETEROCYCLIC PROTEIN KINASE INHIBITORS TOLERO PHARMACEUTICALS INC (US) 2020-09-16 EP disclosed
EP-2734205-B1 HETEROCYCLIC PROTEIN KINASE INHIBITORS TOLERO PHARMACEUTICALS INC (US) 2018-03-21 EP disclosed