SCHEMBL19987306

SCHEMBL19987306

CCc1nc(Cl)nc2c1ncn2[C@@H]1O[C@H](CO)C(C)(COP(=O)(N[C@@H](C)C(=O)OC(C)C)Oc2ccccc2)C1F

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
BTN3A1 O00481 1/20 0.38
NT5E P21589 8/20 0.37
ADORA1 P30542 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19987229 0.91 CYP3A4 (0.41) CYP3A4CYP2C9BTN3A1NT5EADORA1
SCHEMBL19987157 0.87 NT5E (0.44) CYP3A4CYP2C9NT5E
SCHEMBL19987313 0.87 NT5E (0.44) CYP3A4CYP2C9NT5E
SCHEMBL19987159 0.86 CYP3A4 (0.43) CYP3A4CYP2C9BTN3A1NT5E
SCHEMBL19987158 0.84 NT5E (0.53) NT5E
SCHEMBL19987209 0.83 NT5E (0.45) CYP3A4CYP2C9NT5E
SCHEMBL19987203 0.83 NT5E (0.44) CYP3A4CYP2C9NT5E
SCHEMBL19987171 0.83 CYP3A4 (0.43) CYP3A4CYP2C9BTN3A1NT5EADORA1
SCHEMBL19987346 0.82 NT5E (0.40) CYP3A4CYP2C9NT5E
SCHEMBL19987198 0.81 PDE2A (0.46) CYP3A4CYP2C9NT5E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018049535-A1 NUCLEOSIDE ANALOGUES AND METHODS OF USE THEREOF LCB PHARMA INC. (CA) 2018-03-22 WO disclosed