SCHEMBL20004751

SCHEMBL20004751

C/N=C\c1ccc2c3c([nH]c2c1)C(C)(C)c1ccc(OC)cc1C3

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
CA4 P22748 3/20 0.41
CA6 P23280 3/20 0.41
KDM4E B2RXH2 5/20 0.36
MAPT P10636 3/20 0.36
POLB P06746 3/20 0.36
GAA P10253 2/20 0.36
PSMD14 O00487 1/20 0.36
KMT2A Q03164 4/20 0.36
HTR7 P34969 2/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
NISCH Q9Y2I1 1/20 0.35
MAPK10 P53779 1/20 0.34
RIPK1 Q13546 1/20 0.34
DRD2 P14416 1/20 0.34
DRD1 P21728 1/20 0.34
DRD5 P21918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1755993 0.81 CA1 (0.48) CA1CA2CA4CA6KDM4E
SCHEMBL897691 0.78 ALK (0.50) ALK
SCHEMBL21443127 0.77 ALK (0.49) KDM4EMAPTPOLBGAAKMT2A
SCHEMBL896972 0.73 CDK4 (0.46) CA1CA2CA4CA6KDM4E
SCHEMBL897959 0.73 CA1 (0.43) CA1CA2CA4CA6KDM4E
SCHEMBL20004253 0.71 CA1 (0.32) CA1CA2CA4CA6ALK
SCHEMBL23027947 0.70 CA1 (0.45) CA1CA2CA4CA6KDM4E
SCHEMBL897447 0.70 CA1 (0.43) CA1CA2CA4CA6KDM4E
SCHEMBL898273 0.69 CA1 (0.41) CA1CA2CA4CA6KDM4E
SCHEMBL21613391 0.69 CA1 (0.40) CA1CA2CA4CA6HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2975024-B1 TETRACYCLIC COMPOUNDS CHUGAI PHARMACEUTICAL CO LTD (JP) 2018-03-28 EP disclosed