SCHEMBL20004986

SCHEMBL20004986

CC(C)c1ccc(COCc2cccc(I)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.50
TACR1 P25103 2/20 0.50
MRGPRX4 Q96LA9 1/20 0.43
TSHR P16473 1/20 0.39
NFE2L2 Q16236 1/20 0.38
ALOX5 P09917 1/20 0.37
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
NLRP3 Q96P20 1/20 0.37
APP P05067 1/20 0.36
SLC2A1 P11166 1/20 0.36
EGLN1 Q9GZT9 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
THPO P40225 1/20 0.36
RAB9A P51151 1/20 0.36
HIF1A Q16665 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7892498 0.82 IDO1 (0.69) IDO1TACR1TSHRCYP1A2CYP2D6
SCHEMBL22537583 0.82 IDO1 (0.51) IDO1TACR1MRGPRX4TSHRNFE2L2
SCHEMBL13756779 0.81 TSHR (0.62) IDO1TACR1TSHRNFE2L2ALOX5
SCHEMBL9842310 0.81 TSHR (0.62) IDO1TACR1TSHRNFE2L2ALOX5
SCHEMBL15687841 0.81 TSHR (0.62) IDO1TACR1TSHRAPPCYP1A2
SCHEMBL20004351 0.81 IDO1 (0.50) IDO1MRGPRX4
SCHEMBL2293769 0.80 IDO1 (0.68) IDO1TSHRNFE2L2ALOX5RXRA
SCHEMBL5250014 0.79 APP (0.53) IDO1TACR1MRGPRX4APPRAB9A
SCHEMBL4507875 0.79 APP (0.53) IDO1TACR1MRGPRX4APPRAB9A
SCHEMBL29041352 0.79 TSHR (0.65) IDO1TACR1MRGPRX4TSHRRXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3515912-B1 COMPOUNDS FOR USING IN IMAGING AND PARTICULARLY FOR THE DIAGNOSIS OF NEURODEGENERATIVE DISEASES CENTRE NAT RECH SCIENT (FR) 2020-10-14 EP disclosed
WO-2018055316-A1 COMPOUNDS FOR USING IN IMAGING AND PARTICULARLY FOR THE DIAGNOSIS OF NEURODEGENERATIVE DISEASES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2018-03-29 WO disclosed