SCHEMBL20006198

SCHEMBL20006198

CC12CCC3c4ccc(C#N)cc4CCC3C1CC=C2c1cncc(F)c1

nearest known ligand 0.65

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 20/20 0.65
CYP17A1 P05093 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15974275 1.00 AKR1C3 (0.65) AKR1C3CYP17A1
SCHEMBL15974295 0.89 CYP17A1 (0.60) AKR1C3CYP17A1
SCHEMBL20006567 0.89 CYP17A1 (0.60) AKR1C3CYP17A1
SCHEMBL15414510 0.87 CYP17A1 (0.74) AKR1C3CYP17A1
SCHEMBL17597411 0.86 AKR1C3 (0.68) AKR1C3CYP17A1
SCHEMBL17597459 0.85 AKR1C3 (0.69) AKR1C3CYP17A1
SCHEMBL15415077 0.84 AKR1C3 (0.67) AKR1C3CYP17A1
SCHEMBL17597340 0.84 AKR1C3 (0.67) AKR1C3CYP17A1
SCHEMBL17457514 0.83 AKR1C3 (0.62) AKR1C3CYP17A1
SCHEMBL20006531 0.83 AKR1C3 (0.79) AKR1C3CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2958928-B1 ESTRA-1,3,5(10),16-TETRAENE-3-CARBOXAMIDES FOR INHIBITION OF 17.BETA.-HYDROXYSTEROID DEHYDROGENASE (AKR1 C3) Bayer Pharma AG (DE) 2018-03-28 EP disclosed