SCHEMBL20007791

SCHEMBL20007791

O=C(NCc1ccc(F)cc1F)c1cn2c(c(O)c1=O)C(=O)N1C(C2)NOCC2CCCC21

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC22A2 O15244 19/20 0.67
CYP3A4 P08684 1/20 0.62
TMEM97 Q5BJF2 1/20 0.62
ABCG2 Q9UNQ0 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15089841 0.89 SLC22A2 (0.69) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL2679002 0.87 SLC22A2 (0.74) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL29775438 0.87 SLC22A2 (0.74) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL82784 0.87 SLC22A2 (0.74) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL19327604 0.87 SLC22A2 (0.74) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL19739113 0.87 SLC22A2 (0.74) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL30231883 0.87 SLC22A2 (0.74) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL17005316 0.85 SLC22A2 (0.74) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL17923551 0.85 SLC22A2 (0.74) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL18424163 0.85 SLC22A2 (0.74) SLC22A2CYP3A4TMEM97ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3045206-B2 POLYCYCLIC CARBAMOYLPYRIDONE DERIVATIVE HAVING HIV INTEGRASE INHIBITORY ACTIVITY VIIV HEALTHCARE CO (US) 2023-02-15 EP disclosed
EP-3045206-B1 POLYCYCLIC CARBAMOYLPYRIDONE DERIVATIVE HAVING HIV INTEGRASE INHIBITORY ACTIVITY VIIV HEALTHCARE CO (US) 2018-03-28 EP disclosed