SCHEMBL20021148

SCHEMBL20021148

Cc1cc2nc(-c3ccnnc3)ccc2c(-c2ccc3c4c(ccnc24)CCO3)c1C(OC(C)(C)C)C(=O)O

nearest known ligand 0.68

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.68
PSIP1 O75475 1/20 0.37
NR1I2 O75469 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL244981 1.00 CYP3A4 (0.68) CYP3A4PSIP1NR1I2
SCHEMBL15182676 0.94 CYP3A4 (0.59) CYP3A4PSIP1
SCHEMBL246526 0.93 CYP3A4 (0.69) CYP3A4PSIP1NR1I2
SCHEMBL244833 0.92 CYP3A4 (0.75) CYP3A4PSIP1NR1I2
SCHEMBL244314 0.92 CYP3A4 (0.68) CYP3A4PSIP1NR1I2
SCHEMBL251326 0.91 CYP3A4 (0.67) CYP3A4PSIP1NR1I2
SCHEMBL244883 0.91 CYP3A4 (0.69) CYP3A4PSIP1NR1I2
SCHEMBL244974 0.90 CYP3A4 (0.68) CYP3A4PSIP1NR1I2
SCHEMBL245459 0.90 CYP3A4 (0.68) CYP3A4PSIP1NR1I2
SCHEMBL242145 0.89 CYP3A4 (0.72) CYP3A4PSIP1NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588455-B1 2-QUINOLINYL-ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES INC (US) 2018-04-04 EP disclosed