SCHEMBL20021188

SCHEMBL20021188

CCCc1ccc2c(-c3ccc4c5c(ccnc35)CCO4)c([C@H](OC(C)(C)C)C(=O)O)c(C)cc2n1

nearest known ligand 0.69

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.69
PSIP1 O75475 1/20 0.36
MAPK14 Q16539 4/20 0.31
NR1I2 O75469 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL241605 0.94 CYP3A4 (0.69) CYP3A4PSIP1MAPK14NR1I2
SCHEMBL3320041 0.94 CYP3A4 (0.71) CYP3A4PSIP1MAPK14NR1I2
SCHEMBL244246 0.93 CYP3A4 (0.71) CYP3A4PSIP1MAPK14NR1I2
SCHEMBL244245 0.93 CYP3A4 (0.71) CYP3A4PSIP1MAPK14NR1I2
SCHEMBL247066 0.93 CYP3A4 (0.71) CYP3A4PSIP1MAPK14NR1I2
SCHEMBL245707 0.92 CYP3A4 (0.67) CYP3A4PSIP1MAPK14
SCHEMBL245778 0.92 CYP3A4 (0.71) CYP3A4PSIP1MAPK14NR1I2
SCHEMBL245427 0.92 CYP3A4 (0.68) CYP3A4PSIP1NR1I2
SCHEMBL245426 0.92 CYP3A4 (0.68) CYP3A4PSIP1NR1I2
SCHEMBL245035 0.92 CYP3A4 (0.66) CYP3A4PSIP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588455-B1 2-QUINOLINYL-ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES INC (US) 2018-04-04 EP disclosed