SCHEMBL20021215

SCHEMBL20021215

c1cn2ccnc2c(N2CCCC2)n1

nearest known ligand 0.70

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.45
ACKR3 P25106 1/20 0.44
NUDT1 P36639 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7324694 0.82 PIK3R1 (0.55) HTR2CACKR3KDM4EGAA
SCHEMBL5496661 0.82 HTR2C (0.65) HTR2C
SCHEMBL9963421 0.81 PDE10A (0.42) HTR2CACKR3TSHR
Hydrochloric Acid SCHEMBL11172195 0.80 HTR2C (0.61) HTR2C
SCHEMBL2312218 0.80 ACKR3 (0.44) ACKR3KDM4EALDH1A1GLAGAA
SCHEMBL19222166 0.76 GRIA1 (0.43) HTR2C
SCHEMBL17793382 0.73 HTR2C (0.45) HTR2CACKR3
SCHEMBL19468828 0.73 HTR2C (0.45) HTR2CACKR3
SCHEMBL15754793 0.73 ACKR3 (0.46) ACKR3
SCHEMBL15760247 0.73 ACKR3 (0.48) ACKR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3564235-A1 SUBSTITUTED AROMATIC N-HETEROCYCLIC COMPOUNDS AS INHIBITORS OF MITOGEN-ACTIVATED PROTEIN KINASE INTERACTING KINASE 1 (MNK1) AND 2 (MNK2) Northwestern University (US) 2019-11-06 EP disclosed
EP-2925745-B1 CXCR7 ANTAGONISTS CHEMOCENTRYX INC (US) 2018-04-04 EP disclosed