SCHEMBL20037271

SCHEMBL20037271

Cc1nn(-c2ccc(C(F)(F)F)cc2)c(C)c1NC(O)COC(=O)Cn1c(C)cc2ccccc21

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK6 Q92876 6/20 0.59
PRSS1 P07477 1/20 0.59
PRSS2 P07478 1/20 0.59
PRSS3 P35030 1/20 0.59
RXFP1 Q9HBX9 1/20 0.40
P2RX7 Q99572 1/20 0.37
GSR P00390 2/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
KDM4E B2RXH2 2/20 0.36
LMNA P02545 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PPARG P37231 1/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
RAB9A P51151 2/20 0.35
HTT P42858 1/20 0.34
TP53 P04637 1/20 0.34
BRAF P15056 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20037103 0.91 KLK6 (0.64) KLK6PRSS1PRSS2PRSS3MEN1
SCHEMBL20037144 0.86 KLK6 (0.62) KLK6PRSS1PRSS2PRSS3MEN1
SCHEMBL20037280 0.85 KLK6 (0.82) KLK6PRSS1PRSS2PRSS3MEN1
SCHEMBL20037005 0.75 KLK6 (0.89) KLK6PRSS1PRSS2PRSS3MEN1
SCHEMBL20037270 0.75 KLK6 (1.00) KLK6PRSS1PRSS2PRSS3MEN1
SCHEMBL20037221 0.74 KLK6 (0.86) KLK6PRSS1PRSS2PRSS3MEN1
SCHEMBL20037080 0.73 KLK6 (0.82) KLK6PRSS1PRSS2PRSS3MEN1
SCHEMBL20037050 0.73 KLK6 (0.71) KLK6PRSS1PRSS2PRSS3MEN1
SCHEMBL20037182 0.73 KLK6 (0.79) KLK6PRSS1PRSS2PRSS3MEN1
SCHEMBL20037009 0.72 KLK6 (0.73) KLK6PRSS1PRSS2PRSS3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3305781-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN-RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum (DE) 2018-04-11 EP disclosed