SCHEMBL20037587

SCHEMBL20037587

Nc1ccc(NC2CCNCC2)cn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.49
PLK4 O00444 2/20 0.46
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
MAPK1 P28482 1/20 0.39
CDK4 P11802 2/20 0.39
CDK1 P06493 1/20 0.39
CCND1 P24385 1/20 0.39
CDK2 P24941 1/20 0.39
HRH4 Q9H3N8 1/20 0.38
HTR6 P50406 3/20 0.38
CDK6 Q00534 1/20 0.38
CYP1A2 P05177 2/20 0.38
MEN1 O00255 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
KMT2A Q03164 1/20 0.38
USP2 O75604 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17054985 0.84 KIT (0.41) MAPK1MEN1KMT2AALDH1A1HSD17B10
SCHEMBL21606946 0.80 BRD4 (0.46) HRH3PLK4CTSLCTSBCTSS
SCHEMBL7105363 0.80 IKBKB (0.43) HRH3PLK4CTSLCTSBCTSS
SCHEMBL2233319 0.77 PLK4 (0.54) HRH3PLK4CTSLCTSBCTSS
SCHEMBL24529842 0.76 PIK3CA (0.52) CTSLCTSBCTSSCTSKMAPK1
SCHEMBL26330921 0.76 BRD4 (0.47) CTSLCTSBCTSSCTSKCDK4
SCHEMBL28823771 0.76 CHEK1 (0.60) CTSLCTSBCTSSCTSKCHEK1
SCHEMBL31247376 0.76 HDAC1 (0.36) PLK4NOS2
Hydrochloric Acid SCHEMBL25221350 0.75 BRD4 (0.47) CTSLCTSBCTSSCTSKCDK4
Hydrochloric Acid SCHEMBL22031708 0.75 CHEK1 (0.45) HRH3PLK4CTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3305785-A1 PYRIDO[3,4-d]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Teijin Pharma Limited (JP) 2018-04-11 EP disclosed