SCHEMBL20037693

SCHEMBL20037693

O=C1C[C@@H](O)CN1c1ccc(I)nc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.44
RXFP1 Q9HBX9 1/20 0.35
TSHR P16473 2/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
CA5B Q9Y2D0 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
DPP4 P27487 3/20 0.33
NPC1 O15118 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18291570 0.85 HRH3 (0.39) HRH3RXFP1KMT2AMEN1ALDH1A1
SCHEMBL20037471 0.85 HRH3 (0.39) HRH3RXFP1KMT2AMEN1ALDH1A1
SCHEMBL20037438 0.83 HRH3 (0.45) HRH3RXFP1TSHRMAPK1KMT2A
SCHEMBL20037429 0.82 HRH3 (0.44) HRH3TSHRMAPK1KMT2AMEN1
SCHEMBL20037692 0.82 HRH3 (0.44) HRH3TSHRMAPK1KMT2AMEN1
SCHEMBL19302977 0.79 TSHR (0.41) HRH3RXFP1TSHRMAPK1KMT2A
SCHEMBL12407039 0.78 HRH3 (0.42) HRH3RXFP1TSHRMAPK1KMT2A
SCHEMBL12485053 0.78 DPP4 (0.51) HRH3RXFP1KMT2AMEN1ALDH1A1
SCHEMBL20249134 0.78 HRH3 (0.42) HRH3TSHRMAPK1KMT2AMEN1
SCHEMBL20249135 0.78 HRH3 (0.42) HRH3TSHRMAPK1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3305785-A1 PYRIDO[3,4-d]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Teijin Pharma Limited (JP) 2018-04-11 EP disclosed