SCHEMBL20042662

SCHEMBL20042662

Cc1nc(O)c2c(n1)CN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
C5AR1 P21730 1/20 0.39
PARP1 P09874 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
MTOR P42345 1/20 0.38
GPR119 Q8TDV5 1/20 0.37
ESR2 Q92731 1/20 0.36
USP2 O75604 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MKNK1 Q9BUB5 4/20 0.36
DDB1 Q16531 2/20 0.35
CRBN Q96SW2 2/20 0.35
MAPT P10636 1/20 0.35
NR1H2 P55055 1/20 0.34
ADORA1 P30542 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31016562 1.00 C5AR1 (0.39) C5AR1PARP1TNKS2PARP2MTOR
SCHEMBL30776218 0.88 ESR2 (0.45) C5AR1PARP1TNKS2PARP2MTOR
SCHEMBL30776241 0.88 PARP1 (0.47) C5AR1PARP1TNKS2PARP2MTOR
SCHEMBL12706727 0.88 ESR2 (0.45) C5AR1PARP1TNKS2PARP2MTOR
SCHEMBL13250465 0.88 PARP1 (0.47) C5AR1PARP1TNKS2PARP2MTOR
SCHEMBL19357859 0.84 C5AR1 (0.39) C5AR1PARP1TNKS2PARP2MTOR
SCHEMBL20608461 0.84 C5AR1 (0.39) C5AR1PARP1TNKS2PARP2MTOR
SCHEMBL28672930 0.84 POLB (0.39) C5AR1PARP1TNKS2PARP2MTOR
SCHEMBL31016608 0.83 PARP1 (0.37) C5AR1PARP1TNKS2PARP2MTOR
SCHEMBL27270234 0.83 C5AR1 (0.38) C5AR1PARP1TNKS2PARP2MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113727758-A Bicyclic heterocyclic compounds and use thereof 锐新医药公司 2021-11-30 CN disclosed
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed