SCHEMBL20046949

SCHEMBL20046949

O=C1C(C2=C(N3CCN(CCOCCO)CC3)C(=O)c3ccccc3C2=O)=C(N2CCN(CCOCCO)CC2)C(=O)c2ccccc21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC25B P30305 1/20 0.58
CHRM2 P08172 2/20 0.53
ADRA2A P08913 2/20 0.53
DRD2 P14416 2/20 0.53
ADRA2B P18089 2/20 0.53
ADRA2C P18825 2/20 0.53
DRD4 P21917 2/20 0.53
HRH2 P25021 2/20 0.53
HTR2A P28223 2/20 0.53
HTR7 P34969 2/20 0.53
ADRA1A P35348 2/20 0.53
HRH1 P35367 2/20 0.53
DRD3 P35462 2/20 0.53
OPRK1 P41145 2/20 0.53
HTR2B P41595 2/20 0.53
HTR6 P50406 2/20 0.53
KCNH2 Q12809 2/20 0.53
LMNA P02545 2/20 0.53
CHRM4 P08173 1/20 0.53
CYP3A4 P08684 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20046958 0.86 MAPT (0.60) CDC25BDRD2DRD3LMNAKDM4E
SCHEMBL20046775 0.80 NSD2 (0.53) CDC25BDRD2DRD3LMNAMEN1
SCHEMBL20046757 0.77 MAPT (0.67) CDC25BLMNAKDM4EMEN1MAPK1
SCHEMBL22266161 0.75 KCNH2 (0.62) CHRM2ADRA2ADRD2ADRA2BADRA2C
SCHEMBL11104593 0.75 KDM4E (0.52) CDC25BCHRM2ADRA2ADRD2ADRA2B
SCHEMBL17250432 0.74 NSD2 (0.63) CDC25BDRD2DRD4DRD3LMNA
SCHEMBL17250407 0.73 NSD2 (0.67) CDC25BDRD2DRD3LMNAMEN1
SCHEMBL13856939 0.72 NSD2 (0.52) CDC25BCHRM2ADRA2ADRD2ADRA2B
SCHEMBL8250517 0.70 HRH1 (0.68) CDC25BCHRM2ADRA2ADRD2ADRA2B
SCHEMBL8966405 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11459313-B2 Aziridinyl and amino dimeric naphthoquinone compounds and use for acute myeloid leukemia UNIVERSITY OF MARYLAND, BALTIMORE (US) 2022-10-04 US disclosed
US-20200283417-A1 AZIRIDINYL AND AMINO DIMERIC NAPHTHOQUINONE COMPOUNDS AND USE FOR ACUTE MYELOID LEUKEMIA UNIVERSITY OF MARYLAND, BALTIMORE 2020-09-10 US disclosed
US-20200283417-A1 AZIRIDINYL AND AMINO DIMERIC NAPHTHOQUINONE COMPOUNDS AND USE FOR ACUTE MYELOID LEUKEMIA UNIVERSITY OF MARYLAND, BALTIMORE 2020-09-10 US disclosed
WO-2018067842-A1 AZIRIDINYL AND AMINO DIMERIC NAPHTHOQUINONE COMPOUNDS AND USE FOR ACUTE MYELOID LEUKEMIA UNIVERSITY OF MARYLAND, BALTIMORE (US) 2018-04-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200283417-A1 AZIRIDINYL AND AMINO DIMERIC NAPHTHOQUINONE COMPOUNDS AND USE FOR ACUTE MYELOID LEUKEMIA MCL1, NPM1, ABL1 CDC25B 502/4885CHRM2 2212/4885ADRA2A 1766/4885
US-11459313-B2 Aziridinyl and amino dimeric naphthoquinone compounds and use for acute myeloid leukemia MCL1, NPM1, ABL1 CDC25B 502/4885CHRM2 2212/4885ADRA2A 1766/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.