SCHEMBL20051520

SCHEMBL20051520

COc1ccc(Cn2c(C)c(C#N)c(-c3ccc(C#N)cc3)c2C)cc1

nearest known ligand 0.72

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AR P10275 7/20 0.72
GRIN1 Q05586 1/20 0.48
GRIN2B Q13224 1/20 0.48
MAPT P10636 3/20 0.47
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
ALOX15 P16050 1/20 0.47
CYP19A1 P11511 2/20 0.46
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
GAA P10253 2/20 0.43
GFER P55789 1/20 0.43
GLA P06280 1/20 0.43
HPGD P15428 1/20 0.43
PIK3R1 P27986 1/20 0.42
PIK3CA P42336 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6468889 0.91 AR (0.86) ARALDH1A1KDM4ECYP19A1
SCHEMBL24414502 0.87 AR (0.80) ARALDH1A1CYP19A1KMT2AMEN1
SCHEMBL24414597 0.84 AR (0.65) AR
SCHEMBL24411064 0.84 AR (0.76) ARCYP19A1MAOAMAOBGAA
SCHEMBL24411088 0.84 AR (0.76) ARCYP19A1
SCHEMBL21996432 0.84 AR (0.76) ARCYP19A1
SCHEMBL6468792 0.83 AR (0.80) ARGRIN1GRIN2BMAPTALDH1A1
SCHEMBL20051214 0.82 AR (0.72) ARCYP19A1
SCHEMBL6465872 0.82 AR (0.76) ARCYP19A1
SCHEMBL6468062 0.80 AR (1.00) ARMAPTALDH1A1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066545-A1 HETEROCYCLIC COMPOUND 公益財団法人ヒューマンサイエンス振興財団 2018-04-12 WO disclosed