SCHEMBL20052015

SCHEMBL20052015

CCc1ncncc1-c1cccc2[nH]cnc12

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.42
CYP17A1 P05093 3/20 0.36
PARP1 P09874 1/20 0.36
AURKA O14965 1/20 0.34
JAK2 O60674 1/20 0.34
RPS6KA2 Q15349 1/20 0.34
DPP4 P27487 1/20 0.33
ABL1 P00519 1/20 0.33
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL900129 0.81 BRD4 (0.45) BRD4CYP17A1PARP1AURKAJAK2
SCHEMBL20365106 0.79 BRD4 (0.43) BRD4CYP17A1PARP1AURKAJAK2
SCHEMBL20878376 0.76 BRD4 (0.56) BRD4PARP1AURKAJAK2RPS6KA2
SCHEMBL903206 0.74 BRD4 (0.52) BRD4PARP1DPP4ABL1DRD4
SCHEMBL903194 0.72 CYP17A1 (0.50) BRD4CYP17A1
SCHEMBL900109 0.70 CYP17A1 (0.48) BRD4CYP17A1PARP1AURKAJAK2
SCHEMBL27151824 0.70 PARP1 (0.42) BRD4PARP1AURKAJAK2RPS6KA2
SCHEMBL15159073 0.70 SLC22A12 (0.53) BRD4PARP1
SCHEMBL900402 0.69 BRD4 (0.58) BRD4AURKAJAK2RPS6KA2ABL1
SCHEMBL763087 0.69 PARP1 (0.50) BRD4PARP1DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9944619-B2 Compounds for the treatment of HIV GILEAD SCIENCES, INC. (US) 2018-04-17 US disclosed