SCHEMBL20053763

SCHEMBL20053763

C[C@H](N)CC[C@@H](C)NC(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA7 P43166 2/20 0.49
CYP2D6 P10635 1/20 0.44
CTSK P43235 12/20 0.43
CTSS P25774 6/20 0.42
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.40
KMT2A Q03164 1/20 0.40
CA4 P22748 1/20 0.40
CA9 Q16790 1/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23818566 1.00 CA1 (0.49) CA1CA2CA7CYP2D6CTSK
SCHEMBL23818512 1.00 CA1 (0.49) CA1CA2CA7CYP2D6CTSK
SCHEMBL18660900 1.00 CA1 (0.49) CA1CA2CA7CYP2D6CTSK
SCHEMBL2388142 0.85 CA1 (0.51) CA1CA2CA7CYP2D6CTSK
SCHEMBL2389101 0.85 CA1 (0.51) CA1CA2CA7CYP2D6CTSK
SCHEMBL4464374 0.85 CA1 (0.51) CA1CA2CA7CYP2D6CTSK
SCHEMBL23143036 0.84 CA1 (0.50) CA1CA2CA7CYP2D6CTSK
SCHEMBL23143038 0.84 CA1 (0.50) CA1CA2CA7CYP2D6CTSK
SCHEMBL17150713 0.84 CA1 (0.50) CA1CA2CA7CYP2D6CTSK
SCHEMBL86237 0.84 CA1 (0.50) CA1CA2CA7CYP2D6CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9944612-B2 1-phenyl-2-pyridinyl alkyl alcohol derivatives as phosphodiesterase inhibitors CHIESI FARMACEUTICI S.P.A. (IT) 2018-04-17 US disclosed