SCHEMBL20053791

SCHEMBL20053791

CC(=S)c1nnc2cc(C(=O)O)ccn12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 8/20 0.35
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 3/20 0.35
GAA P10253 2/20 0.35
PKM P14618 1/20 0.35
MAPK13 O15264 1/20 0.34
JMJD6 Q6NYC1 1/20 0.33
AKT1 P31749 1/20 0.33
AKT2 P31751 1/20 0.33
HPGD P15428 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
TSHR P16473 1/20 0.32
RAB9A P51151 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
DNMT1 P26358 1/20 0.31
KDM6B O15054 1/20 0.31
TET3 O43151 1/20 0.31
KDM4A O75164 1/20 0.31
BBOX1 O75936 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10378912 0.78 KDM4E (0.40) HCAR3KDM4EALDH1A1GAAPKM
SCHEMBL15907100 0.74 MAPK13 (0.49) HCAR3KDM4EMAPK13JMJD6MEN1
SCHEMBL22958082 0.74 NR4A1 (0.42) HCAR3KDM4EALDH1A1JMJD6HPGD
SCHEMBL17229830 0.74 MAPK13 (0.49) HCAR3MAPK13JMJD6HPGDHCAR2
SCHEMBL15900088 0.74 DNMT1 (0.45) HCAR3KDM4EALDH1A1GAAHPGD
SCHEMBL29119692 0.67 KDM4E (0.50) KDM4EALDH1A1GAAPKMJMJD6
SCHEMBL973778 0.67 TDP1 (0.45) KDM4EALDH1A1GAAPKMAKT1
SCHEMBL9753645 0.65 NPC1 (0.47) KDM4EALDH1A1GAAPKMJMJD6
SCHEMBL30864250 0.65 JMJD6 (0.37) HCAR3KDM4EALDH1A1GAAPKM
SCHEMBL22366513 0.65 TDP1 (0.42) KDM4EALDH1A1GAAAKT1AKT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9944644-B2 Octahydropyrrolopyrroles their preparation and use THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2018-04-17 US disclosed