SCHEMBL20053835

SCHEMBL20053835

CCn1nc(S)c2ccc(F)cc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.43
ADORA2B P29275 2/20 0.43
ESR1 P03372 1/20 0.40
RBP4 P02753 1/20 0.39
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PDE5A O76074 2/20 0.34
ATM Q13315 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
DRD2 P14416 1/20 0.33
SLC6A4 P31645 1/20 0.33
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
HTR6 P50406 1/20 0.33
RPS6KA5 O75582 1/20 0.32
ICMT O60725 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17232702 0.81 ADORA2A (0.62) ADORA2AADORA2BESR1RBP4KDM4E
SCHEMBL24045599 0.80 ADORA2A (0.43) ADORA2AADORA2BESR1RBP4KDM4E
SCHEMBL17229778 0.78 ADORA2A (0.41) ADORA2AADORA2BESR1RBP4KDM4E
SCHEMBL17232744 0.71 ADORA2A (0.62) ADORA2AADORA2BKDM4EMAPTMAPK1
SCHEMBL21334032 0.70 KDM4E (0.41) ADORA2AADORA2BESR1KDM4EMAPT
SCHEMBL31052439 0.70 MAPT (0.41) ADORA2AADORA2BESR1KDM4EMAPT
SCHEMBL15832959 0.70 KDM4E (0.41) ADORA2AADORA2BESR1KDM4EMAPT
SCHEMBL16682174 0.69 ADORA2A (0.65) ADORA2AADORA2BESR1ATMDRD2
SCHEMBL22958099 0.68 MAPT (0.40) ADORA2AADORA2BESR1KDM4EMAPT
SCHEMBL20371659 0.68 MAPT (0.40) ADORA2AADORA2BRBP4KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9944644-B2 Octahydropyrrolopyrroles their preparation and use THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2018-04-17 US disclosed