SCHEMBL20054436

SCHEMBL20054436

O=C(NCc1ncc(CCc2ccc3cc(-c4cnc(CNC(=O)C5CCC(F)(F)CC5)[nH]4)ccc3c2)[nH]1)C1CCC(F)(F)CC1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 9/20 0.51
DYRK1A Q13627 9/20 0.51
WNT1 P04628 7/20 0.41
ABL1 P00519 8/20 0.39
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20221278 0.94 GSK3B (0.47) GSK3BDYRK1AWNT1ABL1HDAC3
SCHEMBL20054480 0.91 GSK3B (0.61) GSK3BDYRK1AWNT1ABL1
SCHEMBL20054419 0.90 GSK3B (0.60) GSK3BDYRK1AWNT1ABL1HDAC3
SCHEMBL20054396 0.83 GSK3B (0.55) GSK3BDYRK1AWNT1ABL1HDAC3
SCHEMBL20054523 0.83 GSK3B (0.53) GSK3BDYRK1AWNT1ABL1HDAC3
SCHEMBL20221566 0.83 GSK3B (0.53) GSK3BDYRK1AWNT1ABL1HDAC3
SCHEMBL20054363 0.82 GSK3B (0.49) GSK3BDYRK1AWNT1ABL1HDAC3
SCHEMBL17918629 0.81 GSK3B (0.51) GSK3BDYRK1AWNT1ABL1HDAC3
SCHEMBL15116562 0.80 GSK3B (0.50) GSK3BDYRK1AWNT1ABL1HDAC3
SCHEMBL19388432 0.80 GSK3B (0.50) GSK3BDYRK1AWNT1ABL1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2802326-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-04-18 EP disclosed