SCHEMBL20054567

SCHEMBL20054567

O=C(NCc1ncc(-c2ccc(-c3ccc4nc(CNC(=O)C5CCC(F)(F)CC5)[nH]c4c3)cc2)[nH]1)C1CCC(F)(F)CC1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 8/20 0.48
DYRK1A Q13627 8/20 0.48
WNT1 P04628 6/20 0.41
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
PDPK1 O15530 2/20 0.38
AAK1 Q2M2I8 1/20 0.37
LMNA P02545 2/20 0.37
CDK9 P50750 1/20 0.36
MELK Q14680 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20054445 1.00 GSK3B (0.48) GSK3BDYRK1AWNT1HDAC3HDAC1
SCHEMBL20054523 0.95 GSK3B (0.53) GSK3BDYRK1AWNT1HDAC3HDAC1
SCHEMBL20221305 0.94 GSK3B (0.44) GSK3BDYRK1AWNT1HDAC3HDAC1
SCHEMBL20054351 0.92 GSK3B (0.43) GSK3BDYRK1AWNT1PDPK1AAK1
SCHEMBL20054393 0.91 GSK3B (0.43) GSK3BDYRK1AWNT1HDAC3HDAC1
SCHEMBL20054417 0.87 GSK3B (0.49) GSK3BDYRK1AWNT1HDAC3HDAC1
SCHEMBL20054480 0.86 GSK3B (0.61) GSK3BDYRK1AWNT1
SCHEMBL20221217 0.83 SMN1; SMN2 (0.35) GSK3BDYRK1AHDAC1AAK1LMNA
SCHEMBL20054419 0.83 GSK3B (0.60) GSK3BDYRK1AWNT1HDAC3HDAC1
SCHEMBL20221552 0.81 SMN1; SMN2 (0.36) GSK3BDYRK1AAAK1MELKSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2802326-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-04-18 EP disclosed