SCHEMBL20054776

SCHEMBL20054776

c1nc(-c2ccc(-c3ccc4cc(-c5c[nH]cn5)ccc4c3)cc2)c[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.36
ESR2 Q92731 4/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
CYP1A1 P04798 1/20 0.36
CYP1B1 Q16678 1/20 0.36
CYP1A2 P05177 3/20 0.34
ACVR1 Q04771 1/20 0.33
NPC1 O15118 4/20 0.33
RAB9A P51151 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 1/20 0.33
THRB P10828 1/20 0.33
KMT2A Q03164 1/20 0.33
HTR2B P41595 1/20 0.33
HTR5A P47898 1/20 0.33
ALDH1A1 P00352 3/20 0.33
HPGD P15428 2/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12647726 0.94 CYP11B1 (0.39) ESR1ESR2CYP11B1CYP11B2CYP1A1
SCHEMBL26259879 0.88 CYP11B1 (0.38) ESR1ESR2CYP11B1CYP11B2CYP1A1
SCHEMBL4526053 0.87 CYP11B1 (0.50) ESR1ESR2CYP11B1CYP11B2CYP1A1
SCHEMBL20054187 0.85 AKT1 (0.30)
SCHEMBL17948025 0.84 CYP11B1 (0.56) CYP11B1CYP11B2CYP1A2SMN1; SMN2CYP2C9
SCHEMBL12647439 0.84 CYP11B1 (0.33) CYP11B1CYP11B2CYP1A1CYP1B1CYP1A2
SCHEMBL17948012 0.84 CYP11B1 (0.42) CYP11B1CYP11B2CYP1A1CYP1B1CYP1A2
SCHEMBL12647819 0.82 CYP11B1 (0.62) CYP11B1CYP11B2CYP1A2SMN1; SMN2CYP2C9
SCHEMBL31546885 0.81 NPC1 (0.53) CYP11B1CYP11B2CYP1A2NPC1RAB9A
SCHEMBL12647870 0.80 CYP11B1 (0.64) CYP11B1CYP11B2CYP1A2SMN1; SMN2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3019196-B1 COMBINATIONS OF HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-06-06 EP disclosed
EP-2802326-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-04-18 EP disclosed