SCHEMBL20064314

SCHEMBL20064314

COc1ccccc1OC1CC(C(=O)O)C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 8/20 0.48
PDE4B Q07343 8/20 0.48
PDE4C Q08493 8/20 0.48
PDE4D Q08499 8/20 0.48
EPHX2 P34913 1/20 0.47
LPAR1 Q92633 1/20 0.46
LPAR5 Q9H1C0 1/20 0.46
POLB P06746 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
KMT2A Q03164 2/20 0.44
HTT P42858 1/20 0.44
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA7 P43166 2/20 0.43
CA9 Q16790 2/20 0.43
CA14 Q9ULX7 2/20 0.43
CA4 P22748 1/20 0.43
LMNA P02545 1/20 0.42
FFAR1 O14842 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21222343 1.00 PDE4A (0.48) PDE4APDE4BPDE4CPDE4DEPHX2
SCHEMBL21222345 1.00 PDE4A (0.48) PDE4APDE4BPDE4CPDE4DEPHX2
SCHEMBL16506986 0.85 PDE4A (0.59) PDE4APDE4BPDE4CPDE4DEPHX2
SCHEMBL21222436 0.85 EPHX2 (0.46) PDE4APDE4BPDE4CPDE4DEPHX2
SCHEMBL20064643 0.85 EPHX2 (0.46) PDE4APDE4BPDE4CPDE4DEPHX2
SCHEMBL21222047 0.83 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL21222420 0.83 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DPOLB
SCHEMBL21222421 0.83 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DPOLB
SCHEMBL20064203 0.83 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL21222267 0.81 SLC6A4 (0.57) EPHX2KMT2AFFAR1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed