SCHEMBL20070537

SCHEMBL20070537

CCOc1ncc(CN2C3CC2CN(C)C3)cc1F

nearest known ligand 0.48

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
RET P07949 17/20 0.48
TLR7 Q9NYK1 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21158876 0.90 RET (0.47) RET
SCHEMBL22031241 0.90 RET (0.50) RET
SCHEMBL20148636 0.88 RET (0.46) RET
SCHEMBL20153155 0.87 RET (0.45) RET
SCHEMBL20070542 0.83 RET (0.45) RET
SCHEMBL22660592 0.82 RET (0.53) RET
SCHEMBL29483142 0.82 RET (0.53) RET
SCHEMBL20154602 0.78 RET (0.49) RETTLR7
SCHEMBL18389829 0.77 KDM4E (0.47) RETTLR7
SCHEMBL20154601 0.77 RET (0.50) RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3753939-A1 SUBSTITUTED PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AS RET KINASE INHIBITORS Array Biopharma Inc. (US) 2020-12-23 EP disclosed
EP-3523301-B1 SUBSTITUTED PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AS RET KINASE INHIBITORS ARRAY BIOPHARMA INC (US) 2020-05-27 EP disclosed
WO-2018071447-A1 SUBSTITUTED PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AS RET KINASE INHIBITORS ANDREWS STEVEN W (US) 2018-04-19 WO disclosed