SCHEMBL20074096

SCHEMBL20074096

CN(C)C(=O)c1ccc(N2CCC[C@@H](CCCN(C)C(=O)C(O)(c3cccc(C4CC4)c3)C(F)(F)F)C2)nc1Cl

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.36
NR1H3 Q13133 2/20 0.36
HSD11B1 P28845 6/20 0.34
ALDH1A1 P00352 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
IDH1 O75874 5/20 0.31
PRCP P42785 1/20 0.31
MAP4K4 O95819 1/20 0.31
GRM2 Q14416 1/20 0.31
DGAT2 Q96PD7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20071835 1.00 NR1H2 (0.36) NR1H2NR1H3HSD11B1ALDH1A1TDP1
SCHEMBL23838196 1.00 NR1H2 (0.36) NR1H2NR1H3HSD11B1ALDH1A1TDP1
SCHEMBL20071914 1.00 NR1H2 (0.36) NR1H2NR1H3HSD11B1ALDH1A1TDP1
SCHEMBL23838164 1.00 NR1H2 (0.36) NR1H2NR1H3HSD11B1ALDH1A1TDP1
SCHEMBL20071913 0.92 NR1H2 (0.40) NR1H2NR1H3TDP1GRM2
SCHEMBL23824826 0.92 NR1H2 (0.40) NR1H2NR1H3TDP1GRM2
SCHEMBL21644330 0.92 NR1H2 (0.40) NR1H2NR1H3TDP1GRM2
SCHEMBL20071909 0.89 NR1H2 (0.35) NR1H2NR1H3HSD11B1ALDH1A1TDP1
SCHEMBL20072157 0.84 NR1H2 (0.41) NR1H2NR1H3ALDH1A1
SCHEMBL20074068 0.84 NR1H2 (0.41) NR1H2NR1H3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018071313-A1 N-ARYL AND N-HETEROARYL PIPERIDINE DERIVATIVES AS LIVER X RECEPTOR BETA AGONISTS, COMPOSITIONS, AND THEIR USE MERCK SHARP & DOHME CORP. (US) 2018-04-19 WO disclosed