SCHEMBL20074329

SCHEMBL20074329

CC(C)Cn1cc(-c2[nH]c3ncnn3c(=O)c2C(C)C)cn1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM5B Q9UGL1 14/20 0.52
KDM5A P29375 2/20 0.45
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38
ACHE P22303 2/20 0.37
SYK P43405 1/20 0.37
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21720927 0.89 KDM5B (0.51) KDM5BKDM5ATSHR
SCHEMBL20074100 0.89 KDM5B (0.53) KDM5BKDM5APRMT5WDR77SYK
SCHEMBL21721867 0.87 KDM5B (0.53) KDM5BKDM5ASYKTSHR
SCHEMBL21681722 0.87 KDM5B (0.54) KDM5BKDM5APRMT5WDR77TSHR
SCHEMBL20074327 0.84 KDM5B (0.55) KDM5BSYK
SCHEMBL21721755 0.84 KDM5B (0.55) KDM5BKDM5ASYK
SCHEMBL21721735 0.84 KDM5B (0.47) KDM5BKDM5ATSHR
SCHEMBL20074247 0.84 KDM5B (0.56) KDM5B
SCHEMBL20074323 0.84 KDM5B (0.56) KDM5B
SCHEMBL21681711 0.83 KDM5B (0.48) KDM5BKDM5APRMT5WDR77ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3525785-B1 KDM5 INHIBITORS MERCK SHARP & DOHME LLC (US) 2025-08-27 EP claimed
US-10975084-B2 KDM5 inhibitors MERCK SHARP & DOHME CORP. (US) 2021-04-13 US claimed
US-20200048258-A1 KDM5 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2020-02-13 US claimed
EP-3525785-B1 KDM5 INHIBITORS MERCK SHARP & DOHME LLC (US) 2025-08-27 EP disclosed
US-10975084-B2 KDM5 inhibitors MERCK SHARP & DOHME CORP. (US) 2021-04-13 US disclosed
US-10975084-B2 KDM5 inhibitors MERCK SHARP & DOHME CORP. (US) 2021-04-13 US disclosed
US-20200048258-A1 KDM5 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2020-02-13 US disclosed
US-20200048258-A1 KDM5 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2020-02-13 US disclosed
WO-2018071283-A1 KDM5 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2018-04-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200048258-A1 KDM5 INHIBITORS KDM5A, KDM5B, KDM5C KDM5B 2/4885KDM5A 1/4885PRMT5 33/4885
US-10975084-B2 KDM5 inhibitors KDM5A, KDM5B, KDM5C KDM5B 2/4885KDM5A 1/4885PRMT5 33/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.