SCHEMBL20074871

SCHEMBL20074871

Cc1c(-c2ccc(C(F)F)cc2)nn(CCO)c1N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC34A1 Q06495 11/20 0.38
ESR1 P03372 2/20 0.38
BRD4 O60885 1/20 0.37
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HDAC6 Q9UBN7 1/20 0.34
KDM1A O60341 1/20 0.33
PIK3CD O00329 1/20 0.33
ABL1 P00519 1/20 0.33
EGFR P00533 1/20 0.33
HCK P08631 1/20 0.33
SRC P12931 1/20 0.33
KDR P35968 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
MTOR P42345 1/20 0.33
PIK3CG P48736 1/20 0.33
EPHB4 P54760 1/20 0.33
PRKDC P78527 1/20 0.33
PI4KB Q9UBF8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20075630 0.84 MEN1 (0.41) ESR1BRD4MEN1KMT2ASRC
SCHEMBL20074870 0.84 SLC34A1 (0.52) SLC34A1
SCHEMBL20074790 0.80 SLC34A1 (0.45) SLC34A1KDM1AMBOAT4
SCHEMBL20074681 0.79 SLC34A1 (0.52) SLC34A1MEN1KMT2ASRC
SCHEMBL27516466 0.78 KDR (0.38) ESR1BRD4MEN1KMT2APIK3CD
SCHEMBL1800673 0.73 SMN1; SMN2 (0.41) ESR1BRD4MEN1KMT2ASRC
SCHEMBL24114814 0.69 SLC34A1 (0.40) SLC34A1KMT2A
SCHEMBL20075511 0.69 SLC34A1 (0.50) SLC34A1HDAC6SRCKDR
SCHEMBL20075186 0.68 SLC34A1 (0.45) SLC34A1KDM1A
SCHEMBL12335146 0.67 CYP1A2 (0.41) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3526212-B1 SUBSTITUTED 6-(1H-PYRAZOL-1-YL)PYRIMIDIN-4-AMINE DERIVATIVES AND USES THEREOF BAYER AG (DE) 2021-12-22 EP disclosed
WO-2018069222-A1 SUBSTITUTED 6-(1H-PYRAZOL-1-YL)PYRIMIDIN-4-AMINE DERIVATIVES AND USES THEREOF BAYER AKTIENGESELLSCHAFT (DE) 2018-04-19 WO disclosed