SCHEMBL20074945

SCHEMBL20074945

Cn1nc(N)c(O)c1-c1ccc(F)cc1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.45
GRM5 P41594 13/20 0.41
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAPK13 O15264 2/20 0.37
MAPK12 P53778 2/20 0.37
MAPK11 Q15759 2/20 0.37
CSNK1D P48730 1/20 0.37
CSNK1E P49674 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20075564 0.82 GRM5 (0.47) MAPK14GRM5LMNASMN1; SMN2
SCHEMBL20075418 0.81 MAPK14 (0.44) MAPK14GRM5KDM4EALDH1A1LMNA
SCHEMBL25435704 0.79 MAPK14 (0.43) MAPK14GRM5KDM4EALDH1A1LMNA
SCHEMBL20550958 0.79 KMT2A (0.43) MAPK14GRM5LMNA
SCHEMBL20074942 0.78 SLC34A1 (0.45) MAPK14GRM5KDM4EALDH1A1LMNA
SCHEMBL20075536 0.78 SLC34A1 (0.46) MAPK14
SCHEMBL20075467 0.78 NSD2 (0.45) HTT
SCHEMBL20075477 0.77 MAPK14 (0.59) MAPK14KDM4EALDH1A1LMNAHTT
SCHEMBL21711412 0.77 MAPK14 (0.41) MAPK14GRM5KDM4EALDH1A1LMNA
SCHEMBL20075377 0.77 ADORA2A (0.47) MAPK14KDM4EALDH1A1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069222-A1 SUBSTITUTED 6-(1H-PYRAZOL-1-YL)PYRIMIDIN-4-AMINE DERIVATIVES AND USES THEREOF BAYER AKTIENGESELLSCHAFT (DE) 2018-04-19 WO disclosed