SCHEMBL20076210

SCHEMBL20076210

CC(C)(Cn1ccc(-c2ccc(C#N)c(Cl)c2)n1)NC(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AR P10275 18/20 0.49
AAK1 Q2M2I8 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20046759 0.83 AR (0.65) ARAAK1
SCHEMBL29855799 0.83 AR (0.65) ARAAK1
SCHEMBL31466678 0.83 AR (0.65) ARAAK1
SCHEMBL28440709 0.78 AR (0.45) AR
SCHEMBL20076215 0.78 AR (0.48) AR
SCHEMBL21758951 0.78 AR (0.74) AR
SCHEMBL33526594 0.76 LATS1 (0.35) AAK1
SCHEMBL24652604 0.76 AR (0.47) AR
SCHEMBL24652527 0.76 AR (0.56) AR
SCHEMBL22047519 0.74 AR (0.55) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3660004-B1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF ANDROGEN RECEPTOR ARVINAS OPERATIONS INC (US) 2023-02-22 EP disclosed
EP-3660004-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF ANDROGEN RECEPTOR Arvinas Operations, Inc. (US) 2020-06-03 EP disclosed
WO-2018071606-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF ANDROGEN RECEPTOR Arvinas, Inc. (US) 2018-04-19 WO disclosed