SCHEMBL20084464

SCHEMBL20084464

CNNc1cnc(Oc2c(F)cccc2F)cc1C

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GCK P35557 11/20 0.43
RXRB P28702 2/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ORAI1 Q96D31 1/20 0.32
KDR P35968 2/20 0.32
MAPK14 Q16539 1/20 0.32
TNNI3K Q59H18 1/20 0.32
BRAF P15056 1/20 0.32
SCN8A Q9UQD0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20085248 0.86 MEN1 (0.48) GCKRXRBNPC1RAB9ASMN1; SMN2
SCHEMBL18330558 0.84 GCK (0.41) GCKRXRBNPC1RAB9ASMN1; SMN2
SCHEMBL31221536 0.84 GCK (0.41) GCKRXRBNPC1RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL31221545 0.83 GCK (0.40) GCKRXRBNPC1RAB9ASMN1; SMN2
SCHEMBL20084951 0.81 GCK (0.39) GCKRXRBNPC1RAB9ASMN1; SMN2
SCHEMBL20084783 0.81 GCK (0.46) GCKRXRBSMN1; SMN2MEN1KMT2A
SCHEMBL21971949 0.80 GCK (0.38) GCKNPC1RAB9ASMN1; SMN2MEN1
SCHEMBL18332197 0.80 GCK (0.45) GCKRXRBSMN1; SMN2MEN1KMT2A
SCHEMBL18331768 0.80 MEN1 (0.42) GCKSMN1; SMN2MEN1KMT2A
SCHEMBL20084824 0.79 GCK (0.37) GCKRXRBNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3312172-B1 AMINOPYRAZOLE DERIVATIVES USEFUL AS SRC KINASE INHIBITORS CHUGAI PHARMACEUTICAL CO LTD (JP) 2020-05-06 EP disclosed
EP-3312172-A1 AMINOPYRAZOLE DERIVATIVES Chugai Seiyaku Kabushiki Kaisha (JP) 2018-04-25 EP disclosed