SCHEMBL20103140

SCHEMBL20103140

CC#Cc1cncc(C)n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.33
OGA O60502 1/20 0.32
PIM1 P11309 1/20 0.32
PIM3 Q86V86 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TP53 P04637 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
PKM P14618 1/20 0.31
HPGD P15428 1/20 0.31
ALOX15 P16050 1/20 0.31
CYP2C19 P33261 1/20 0.31
THPO P40225 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31014841 0.78 GRM5 (0.35) GRM5OGAKDM4EMEN1NPC1
SCHEMBL28222619 0.78 GRM5 (0.35) GRM5OGAKDM4EMEN1NPC1
SCHEMBL15871771 0.74
SCHEMBL2632677 0.74
SCHEMBL29955352 0.71
SCHEMBL25429171 0.71 CYP11B1 (0.34) GRM5ALDH1A1CYP1A2RAB9ACYP11B1
SCHEMBL110425 0.71
Ammonia Solution, Strong SCHEMBL28213058 0.68
SCHEMBL23075939 0.68 GRM5 (0.62) GRM5KDM4EMEN1NPC1ALDH1A1
SCHEMBL17066349 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081276-A1 COMPOUNDS TESARO, INC. (US) 2018-05-03 WO disclosed