SCHEMBL20108403

SCHEMBL20108403

COC(=O)c1sc(-c2cnc3cc(Cl)ccn23)cc1OC(C)c1ccccc1C(F)(F)F

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NEK2 P51955 4/20 0.58
FLT3 P36888 1/20 0.58
PLK1 P53350 16/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20108106 0.89 NEK2 (0.57) NEK2FLT3PLK1
SCHEMBL20108284 0.82 NEK2 (0.87) NEK2FLT3PLK1
SCHEMBL2502631 0.82 PLK1 (0.65) NEK2FLT3PLK1
SCHEMBL2523731 0.81 PLK1 (0.77) NEK2FLT3PLK1
SCHEMBL1374710 0.81 PLK1 (0.82) PLK1
SCHEMBL2504909 0.78 PLK1 (0.62) PLK1
SCHEMBL2503660 0.77 PLK1 (0.77) PLK1
SCHEMBL1373276 0.77 PLK1 (0.77) NEK2FLT3PLK1
SCHEMBL2502984 0.75 PLK1 (0.67) PLK1
SCHEMBL2495256 0.75 PLK1 (0.84) PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081719-A1 SMALL MOLECULE INHIBITORS OF NEK2 AND USES THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2018-05-03 WO disclosed