SCHEMBL2011197

SCHEMBL2011197

C1=CN=C1.Cc1ccc(S(=O)(=O)Oc2ccc(Br)nc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
ALDH1A1 P00352 5/20 0.38
MAPT P10636 3/20 0.38
CA12 O43570 2/20 0.38
CA2 P00918 2/20 0.38
HTT P42858 2/20 0.38
PPARG P37231 1/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
NPSR1 Q6W5P4 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
ENPP3 O14638 2/20 0.38
ENPP1 P22413 2/20 0.38
ENPP2 Q13822 2/20 0.38
HPGD P15428 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1979376 0.93 MEN1 (0.47) MEN1KMT2AALDH1A1MAPTCA12
SCHEMBL10684102 0.78 MEN1 (0.49) MEN1KMT2AALDH1A1MAPTCA12
SCHEMBL9852204 0.74 MEN1 (0.60) MEN1KMT2AALDH1A1MAPTCA12
SCHEMBL4126086 0.74 MEN1 (0.60) MEN1KMT2AALDH1A1MAPTCA12
SCHEMBL18179825 0.74 MEN1 (0.60) MEN1KMT2AALDH1A1MAPTCA12
SCHEMBL5255332 0.73 KMT2A (0.45) MEN1KMT2AALDH1A1MAPTCA12
SCHEMBL31637724 0.73 CA12 (0.49) ALDH1A1CA12HPGD
SCHEMBL4195648 0.73 MEN1 (0.53) MEN1KMT2AALDH1A1MAPTCA12
SCHEMBL18359536 0.73 MEN1 (0.53) MEN1KMT2AALDH1A1MAPTCA12
SCHEMBL10678544 0.72 KMT2A (0.47) MEN1KMT2AALDH1A1MAPTCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011072064-A1 S PIRO [CHROMAN - 4, 4 ' - IMIDAZOL] ONES AS BETA - SECRETASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2011-06-16 WO disclosed