SCHEMBL20115918

SCHEMBL20115918

FC(F)(F)Oc1ccc(C#CCC=Cc2ccc(OC(F)(F)F)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.42
GRIK2 Q13002 1/20 0.42
MAOB P27338 1/20 0.39
AOC3 Q16853 1/20 0.39
ACACB O00763 1/20 0.38
CYP2D6 P10635 1/20 0.37
PIM1 P11309 1/20 0.35
PIM2 Q9P1W9 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HRH3 Q9Y5N1 1/20 0.33
CHRNB2 P17787 2/20 0.33
CHRNB4 P30926 2/20 0.33
CHRNA3 P32297 2/20 0.33
CHRNA7 P36544 2/20 0.33
CHRNA4 P43681 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2091009 0.80 GRIK1 (0.48) GRIK1GRIK2MAOBAOC3CYP2D6
SCHEMBL2091007 0.80 GRIK1 (0.48) GRIK1GRIK2MAOBAOC3CYP2D6
SCHEMBL16841023 0.77 ACACB (0.44) MAOBAOC3ACACBFFAR1NOTUM
SCHEMBL19599384 0.76 ACACB (0.42) MAOBAOC3ACACBNOTUMPTGER4
SCHEMBL13790221 0.74 CYP2D6 (0.50) GRIK1GRIK2MAOBAOC3CYP2D6
SCHEMBL4078920 0.74 GRIK1 (0.51) GRIK1GRIK2MAOBAOC3CYP2D6
SCHEMBL4078921 0.74 GRIK1 (0.51) GRIK1GRIK2MAOBAOC3CYP2D6
SCHEMBL1065335 0.74 ACACB (0.43) MAOBAOC3ACACBFFAR1NOTUM
SCHEMBL74114 0.74 GRIK1 (0.48) GRIK1GRIK2MAOBAOC3CYP2D6
SCHEMBL80921 0.74 ACACB (0.46) MAOBAOC3ACACBHRH3FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2870218-B1 BIMESOGENIC COMPOUNDS AND MESOGENIC MEDIA MERCK PATENT GMBH (DE) 2018-05-02 EP disclosed