SCHEMBL20116573

SCHEMBL20116573

CCn1nc(C)c2ccc(C)cc21

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.67
ADORA2B P29275 3/20 0.67
KMO O15229 1/20 0.43
ESR1 P03372 1/20 0.43
SLC22A12 Q96S37 9/20 0.42
GLS O94925 1/20 0.41
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KDM4C Q9H3R0 1/20 0.37
KHK P50053 1/20 0.37
PTGER3 P43115 1/20 0.36
GRM4 Q14833 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26373753 0.82 ADORA2A (0.49) ADORA2AADORA2BKMOESR1LMNA
SCHEMBL16158006 0.82 ADORA2A (0.49) ADORA2AADORA2BESR1LMNAKDM4C
SCHEMBL14910374 0.82 ADORA2A (0.62) ADORA2AADORA2BKMOESR1SLC22A12
SCHEMBL18853871 0.82 ESR1 (0.63) ADORA2AADORA2BKMOESR1SLC22A12
SCHEMBL17232702 0.82 ADORA2A (0.62) ADORA2AADORA2BKMOESR1SLC22A12
SCHEMBL2144945 0.82 ADORA2A (0.62) ADORA2AADORA2BKMOESR1SLC22A12
SCHEMBL14752235 0.82 ADORA2A (0.62) ADORA2AADORA2BKMOESR1SLC22A12
SCHEMBL26373686 0.80 ADORA2A (0.59) ADORA2AADORA2BKMOESR1SLC22A12
SCHEMBL26997295 0.80 ADORA2A (0.59) ADORA2AADORA2BKMOESR1SLC22A12
SCHEMBL14752738 0.78 ADORA2A (0.46) ADORA2AADORA2BKMOSLC22A12GLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019209948-A9 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-01-02 WO disclosed
WO-2019018795-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2019-01-24 WO disclosed
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed