SCHEMBL20116638

SCHEMBL20116638

CCOc1ccc(-c2noc(C3CCN(C(=O)C4CCC(c5ccccc5)N4)CC3)n2)cc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.51
HTT P42858 2/20 0.51
MEN1 O00255 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
KMT2A Q03164 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
SMO Q99835 3/20 0.49
TLR9 Q9NR96 3/20 0.46
TLR8 Q9NR97 3/20 0.46
TLR7 Q9NYK1 3/20 0.46
LMNA P02545 2/20 0.46
USP2 O75604 1/20 0.46
EPHX2 P34913 2/20 0.44
NPC1 O15118 1/20 0.43
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20676406 1.00 TSHR (0.51) TSHRHTTMEN1CYP3A4CYP2C9
SCHEMBL20117108 1.00 TSHR (0.51) TSHRHTTMEN1CYP3A4CYP2C9
SCHEMBL20116587 1.00 TSHR (0.51) TSHRHTTMEN1CYP3A4CYP2C9
SCHEMBL22357786 0.88 HTT (0.50) TSHRHTTMEN1CYP3A4CYP2C9
SCHEMBL21609973 0.83 SMO (0.55) TSHRHTTMEN1CYP3A4CYP2C9
SCHEMBL20660679 0.83 SMO (0.49) TSHRHTTMEN1CYP3A4CYP2C9
SCHEMBL22357969 0.82 HTT (0.55) TSHRHTTMEN1CYP3A4CYP2C9
SCHEMBL22357775 0.82 SMO (0.55) TSHRHTTMEN1CYP3A4CYP2C9
SCHEMBL20116297 0.81 EPHX2 (0.69) TSHRHTTMEN1CYP3A4CYP2C9
SCHEMBL22358183 0.81 HTT (0.56) TSHRHTTMEN1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed