SCHEMBL20117864

SCHEMBL20117864

C1=CC(c2ccc[nH]2)=CNC1

nearest known ligand 0.30

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.30
KDR P35968 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7069184 0.71 AURKA (0.31) AURKAKDR
SCHEMBL630634 0.65 HDAC6 (0.41) AURKAKDR
Hydrochloric Acid SCHEMBL7988951 0.63 HDAC6 (0.40) AURKAKDR
SCHEMBL15828094 0.62 NISCH (0.39)
SCHEMBL3631373 0.60
SCHEMBL3873207 0.59 MEN1 (0.31) AURKAKDR
SCHEMBL2968451 0.59 AURKA (0.31) AURKAKDR
SCHEMBL9419852 0.59 HDAC6 (0.57) AURKAKDR
SCHEMBL20077863 0.58
SCHEMBL18821909 0.57 HDAC6 (0.45) AURKAKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081814-A1 GRP94 SELECTIVE INHIBITORS AND USES THEREOF UNIVERSITY OF KANSAS (US) 2018-05-03 WO disclosed