SCHEMBL20117878

SCHEMBL20117878

NC(=O)c1ccc(-n2cccc2-c2ccccc2Cl)cc1NC1CCCCC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90B1 P14625 2/20 0.50
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA3 P07451 2/20 0.45
CA6 P23280 2/20 0.45
CA7 P43166 2/20 0.45
CA5B Q9Y2D0 2/20 0.45
HSP90AA1 P07900 10/20 0.44
CNR1 P21554 3/20 0.39
JAK2 O60674 2/20 0.39
CNR2 P34972 1/20 0.39
TP53 P04637 1/20 0.39
HSP90AB1 P08238 2/20 0.39
TRAP1 Q12931 1/20 0.39
CISD1 Q9NZ45 1/20 0.39
CA12 O43570 1/20 0.39
CA4 P22748 1/20 0.39
CA9 Q16790 1/20 0.39
CA13 Q8N1Q1 1/20 0.39
CA14 Q9ULX7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20117877 0.91 HSP90B1 (0.61) HSP90B1HSP90AA1HSP90AB1
SCHEMBL20117844 0.88 HSP90B1 (0.50) HSP90B1HSP90AA1CNR1TP53HSP90AB1
SCHEMBL20117784 0.86 HSP90B1 (0.53) HSP90B1CA1CA2CA3CA6
SCHEMBL20117783 0.85 HSP90B1 (0.49) HSP90B1CA1CA2CA3CA6
SCHEMBL20117775 0.83 HSP90B1 (0.47) HSP90B1CA1CA2CA3CA6
SCHEMBL20117712 0.82 HSP90B1 (0.69) HSP90B1CA1CA2CA3CA6
SCHEMBL20117982 0.82 HSP90B1 (0.49) HSP90B1HSP90AA1JAK2JAK1TYK2
SCHEMBL20117777 0.81 HSP90B1 (0.49) HSP90B1CA1CA2CA3CA6
SCHEMBL20117958 0.81 HSP90B1 (0.49) HSP90B1HSP90AA1JAK2HSP90AB1TRAP1
SCHEMBL20117843 0.80 HSP90B1 (0.61) HSP90B1HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081814-A1 GRP94 SELECTIVE INHIBITORS AND USES THEREOF UNIVERSITY OF KANSAS (US) 2018-05-03 WO disclosed