SCHEMBL20118238

SCHEMBL20118238

O=C(N[C@H]1CC[C@@]2(CC1)NC(=O)N(c1ccccc1Cl)C2=O)c1cnn2cccnc12

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 2/20 0.51
JAK1 P23458 1/20 0.51
TYK2 P29597 1/20 0.51
JAK3 P52333 1/20 0.51
TNKS O95271 1/20 0.51
KDM4E B2RXH2 2/20 0.50
HSD17B10 Q99714 2/20 0.50
PKM P14618 1/20 0.50
HSD11B1 P28845 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
IRAK4 Q9NWZ3 11/20 0.44
SYK P43405 2/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
NLRP3 Q96P20 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20118064 1.00 JAK2 (0.51) JAK2JAK1TYK2JAK3TNKS
SCHEMBL18208212 0.84 JAK2 (0.52) JAK2JAK1TYK2JAK3TNKS
SCHEMBL18208215 0.84 JAK2 (0.52) JAK2JAK1TYK2JAK3TNKS
SCHEMBL18208122 0.78 KDM4E (0.50) JAK2JAK1TYK2JAK3TNKS
SCHEMBL18208125 0.78 KDM4E (0.50) JAK2JAK1TYK2JAK3TNKS
SCHEMBL18208937 0.75 TNKS (0.55) TNKSKDM4EHSD17B10PKMHSD11B1
SCHEMBL18208934 0.75 TNKS (0.55) TNKSKDM4EHSD17B10PKMHSD11B1
SCHEMBL18208403 0.74 IRAK4 (0.51) JAK2JAK1TYK2JAK3TNKS
SCHEMBL18208401 0.74 IRAK4 (0.51) JAK2JAK1TYK2JAK3TNKS
SCHEMBL22947094 0.74 KDM4E (0.67) TNKSKDM4EHSD17B10HSD11B1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078009-A1 AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed