SCHEMBL20121533

SCHEMBL20121533

Cc1ccc(Nc2c(-c3ccc(F)cc3)nc3n2CCN(C2OC2C(C)(C)N=[N+]=[N-])C3(C)C)cc1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 10/20 0.49
CYP3A4 P08684 1/20 0.46
MAPT P10636 4/20 0.32
GAA P10253 2/20 0.32
TP53 P04637 1/20 0.31
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15313616 0.78 KCNH2 (0.70) KCNH2CYP3A4MAPTGAATP53
SCHEMBL12781793 0.72 KCNH2 (0.79) KCNH2CYP3A4MAPTGAATP53
SCHEMBL998967 0.71 KCNH2 (0.93) KCNH2CYP3A4MAPTGAATP53
SCHEMBL1051379 0.70 KCNH2 (0.67) KCNH2CYP3A4TP53
SCHEMBL1051946 0.70 KCNH2 (0.55) KCNH2CYP3A4MAPTGAATP53
SCHEMBL998969 0.69 KCNH2 (0.60) KCNH2CYP3A4MAPTGAATP53
SCHEMBL1050138 0.68 KCNH2 (0.93) KCNH2CYP3A4MAPTGAATP53
SCHEMBL15313628 0.68 KCNH2 (0.93) KCNH2CYP3A4MAPTGAATP53
SCHEMBL12845804 0.67 KCNH2 (0.67) KCNH2CYP3A4MAPTGAATP53
SCHEMBL2068986 0.67 KCNH2 (1.00) KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed